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药物发现合肥科生景肽生物科技有限公司是一家专注于肽类药物发现与创新技术服务的高新技术企业。创始团队来自于清华大学和中国科学技术大学,管理团队具备丰富的创新药物研发和技术服务工作经验。
DOTA-[Tyr3]-Octreotide
DOTA-conjugated somatostatin analog for labeling with radiometals such as gallium-67 or gallium-68, indium-111, and yttrium-90. DOTA-TATE is a useful tool in receptor-mediated tumor imaging and peptide receptor-targeted radionuclide therapy.
序列: DOTA-DPhe-Cys-Tyr-DTrp-Lys-Thr-Cys-Thr-ol (trifluoroacetate salt)(Cys2 and 7 bridge)
单字母序列: DOTA-fCYwKTCT-ol (C2&C7 bridge)
参考文献:
L.Kolby et al., Br. J. Cancer, 93, 1144 (2005)
R.Valkema et al., J. Nucl. Med., 46, 83S (2005)
M.de Jong et al., J. Nucl. Med., 46, 13S (2005)
W.A.Breeman et al., Eur. J. Nucl. Med. Mol. Imaging, 30, 917 (2003)
A.Capello et al., Cancer Biother. Radiopharm., 18, 761 (2003)
Chinol, M. et al. Semin. Nucl. Med. 32,141(2002)
De Jong, M. et al. Semin Nucl. Med. 32,133(2002)
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胃肠道疾病相关
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